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My Cart> Small Molecule Compounds > Inhibitors & Antagonists & Agonists > GPCR & G Protein > GW-842166CAS：666260-75-9
Molecular Formula：C18H17Cl2F3N4O2
Molecular Weight：449.25
Storage：Powder:-20℃，2 years;Insolvent(Mother Liquid):-20℃，6 months;-80℃，1 year
Purity：≥98%
Appearance：White to off-white Solid
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| CAS | 666260-75-9 |
| Name | GW-842166 |
| Molecular Formula | C18H17Cl2F3N4O2 |
| Molecular Weight | 449.25 |
| Solubility | Soluble in DMSO ≥1mg/mL(Need ultrasonic) |
| Purity | ≥98% |
| Appearance | White to off-white Solid |
| Storage | Powder:-20℃，2 years;Insolvent(Mother Liquid):-20℃，6 months;-80℃，1 year |
| EC | EINECS 200-258-5 |
| SMILES | ClC1=CC(Cl)=C(NC2=NC=C(C(NCC3CCOCC3)=O)C(C(F)(F)F)=N2)C=C1 |
| Target Point | Cannabinoid Receptor |
| Passage | GPCR & G Protein;Neuronal Signaling |
| Background | GW-842166 is a potent and selective cannabinoid receptor 2 activator. |
| Biological Activity | GW842166X是有效，选择性的 cannabinoid receptor 2 激活剂，IC50 值为63 nM。[1] |
| IC50 | 63nM(human CB2);91nM(rat CB2)[1] |
| Data Literature Source | [1]. Giblin GM，et al. Discovery of 2-[(2，4-dichlorophenyl)amino]-N-[(tetrahydro- 2H-pyran-4-yl)methyl]-4-(trifluoromethyl)- 5-pyrimidinecarboxamide，a selective CB2 receptor agonist for the treatment of inflammatory pain. J Med Chem. 2007 May 31;50(11):2597-600 |
| Unit | Bottle |
| Specification | 5mg 10mg |
Remark：These protocols are for reference only. Solarbio does not independently validate these methods.
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1. The products are all for scientific research use only. Do not use it for medical, clinical diagnosis or treatment, food and cosmetics, etc. Do not store them in ordinary residential areas.
2. For your safety and health, please wear laboratory clothes, disposable gloves and masks.
3. The experimental results may be affected by many factors, after-sale service is limited to the product itself and does not involve other compensation.
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