Mozavaptan
Cat.No:IM2510 Solarbio
CAS:137975-06-5
Molecular Formula:C27H29N3O2
Molecular Weight:427.54
Storage:Powder:2-8℃,2 years
Purity:≥98%
Appearance:White to off-white Solid
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MozavaptanCAS:137975-06-5
Molecular Formula:C27H29N3O2
Molecular Weight:427.54
Storage:Powder:2-8℃,2 years
Purity:≥98%
Appearance:White to off-white Solid
Qty:
Size:
CAS | 137975-06-5 |
Name | Mozavaptan |
Molecular Formula | C27H29N3O2 |
Molecular Weight | 427.54 |
Solubility | Soluble in DMSO ≥0.1mg/mL(Need ultrasonic) |
Purity | ≥98% |
Appearance | White to off-white Solid |
Storage | Powder:2-8℃,2 years |
EC | EINECS 1312995-182-4 |
MDL | MFCD00908918 |
SMILES | CC1=CC=CC=C1C(NC2=CC=C(C(N3C(C=CC=C4)=C4C(N(C)C)CCC3)=O)C=C2)=O |
Target Point | Vasopressin Receptor |
Passage | GPCR & G Protein |
Background | Mozavaptan is a vasopressin V2 receptor antagonist. |
Biological Activity | Mozavaptan (OPC31260)是有口服活性的非肽阴道加压素(vasopressin)V2受体拮抗剂,其IC50值为14nM。[1] |
IC50 | 14nM(vasopressin receptor)[1] |
Data Literature Source | [1]. Yamamura Y,et al. Characterization of a novel aquaretic agent,OPC-31260,as an orally effective,nonpeptide vasopressin V2 receptor antagonist. Br J Pharmacol. 1992 Apr;105(4):787-91 |
Unit | Bottle |
Specification | 5mg 10mg |
Remark:These protocols are for reference only. Solarbio does not independently validate these methods.
Note:
1. The products are all for scientific research use only. Do not use it for medical, clinical diagnosis or treatment, food and cosmetics, etc. Do not store them in ordinary residential areas.
2. For your safety and health, please wear laboratory clothes, disposable gloves and masks.
3. The experimental results may be affected by many factors, after-sale service is limited to the product itself and does not involve other compensation.
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