Your Position: Home > Small Molecule Compounds > Inhibitors & Antagonists & Agonists > GPCR & G Protein > Proxyphylline

Proxyphylline

Manual Download

Cat.No：IP3190 Solarbio

CAS：603-00-9

Molecular Formula：C₁₀H₁₄N₄O₃

Molecular Weight：238.24

Storage：Powder:2-8℃，2 years;Insolvent(Mother Liquid):-20℃，6 months;-80℃，1 year

Purity：≥98%

Appearance：White to off-white Solid

Qty：

Size：

Add to cart

Product Information Experimental Images Related Products Related Paper Technical Q&A

Product Information

CAS	603-00-9
Name	Proxyphylline
Molecular Formula	C₁₀H₁₄N₄O₃
Molecular Weight	238.24
Solubility	Soluble in DMSO ≥2mg/mL(Need ultrasonic)
Purity	≥98%
Appearance	White to off-white Solid
Storage	Powder:2-8℃，2 years;Insolvent(Mother Liquid):-20℃，6 months;-80℃，1 year
EC	EINECS 210-028-7
MDL	MFCD00022833
SMILES	O=C(N1C)N(C)C2=C(N(CC(O)C)C=N2)C1=O
InChIKey	KYHQZNGJUGFTGR-UHFFFAOYSA-N
InChI	InChI=1S/C10H14N4O3/c1-6(15)4-14-5-11-8-7(14)9(16)13(3)10(17)12(8)2/h5-6,15H,4H2,1-3H3
PubChem CID	4977
Target Point	Adenosine Receptor
Passage	GPCR & G Protein
Background	It can selectively antagonize A1 adenosine receptors.
Biological Activity	Proxyphylline是一种甲基黄嘌呤衍生物，临床上作为心脏兴奋剂，血管扩张剂和支气管扩张剂使用。[1-3]
Data Literature Source	[1]. Takeda K，et al. Effects of aminophylline，proxyphylline and a proxyphylline-Melilotus extract-rutin mixture(theoesberiven) on the heart and the coronary circulation. Jpn J Pharmacol. 1977 Oct;27(5):709-20. [2]. Kukovetz WR，et al. Overadditive synergism between theophylline，diprophylline and proxyphylline in tracheal smooth muscle relaxation. Arzneimittelforschung. 1983;33(10):1450-4. [3]. Rasmussen FV，et al. Pharmacokinetics and bronchodilatory effect of proxyphylline and theophylline. Eur J Respir Dis. 1984 Jan;65(1):20-7
Unit	Bottle
Specification	500mg 1g

Remark：These protocols are for reference only. Solarbio does not independently validate these methods.

Note：

1. The products are all for scientific research use only. Do not use it for medical, clinical diagnosis or treatment, food and cosmetics, etc. Do not store them in ordinary residential areas.

2. For your safety and health, please wear laboratory clothes, disposable gloves and masks.

3. The experimental results may be affected by many factors, after-sale service is limited to the product itself and does not involve other compensation.