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My Cart> Small Molecule Compounds > Inhibitors & Antagonists & Agonists > Metabolic Enzyme & Protease > SulfaphenazoleCAS：526-08-9
Molecular Formula：C15H14N4O2S
Molecular Weight：314.36
Storage：Powder:2-8℃，2 years;Insolvent(Mother Liquid):-20℃，6 months;-80℃，1 year
Purity：≥98%
Appearance：White to yellow Solid
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| CAS | 526-08-9 |
| Name | Sulfaphenazole |
| Molecular Formula | C15H14N4O2S |
| Molecular Weight | 314.36 |
| Solubility | Soluble in DMSO |
| Purity | ≥98% |
| Appearance | White to yellow Solid |
| Storage | Powder:2-8℃，2 years;Insolvent(Mother Liquid):-20℃，6 months;-80℃，1 year |
| EC | EINECS 208-384-3 |
| MDL | MFCD00057226 |
| SMILES | O=S(C1=CC=C(N)C=C1)(NC2=CC=NN2C3=CC=CC=C3)=O |
| InChIKey | QWCJHSGMANYXCW-UHFFFAOYSA-N |
| InChI | InChI=1S/C15H14N4O2S/c16-12-6-8-14(9-7-12)22(20,21)18-15-10-11-17-19(15)13-4-2-1-3-5-13/h1-11,18H,16H2 |
| PubChem CID | 5335 |
| Target Point | CYP2C9 |
| Passage | Metabolic Enzyme&Protease |
| Background | It is a specific inhibitor of CYP2C9. |
| Biological Activity | Sulfaphenazole (Depocid, Depotsulfonamide, Plisulfan, Raziosulfa) is an inhibitor of CYP2C9 with Ki value of 0.3 μM and demonstrates at least 100-fold selectivity over other CYP450 isoforms (Ki values of 63 and 29 μM for CYP2C8 and CYP2C18, respectively, and no activity at CYP1A1, CYP1A2, CYP3A4, CYP2C19).[1-2] |
| Data Literature Source | [1] Jeon JH，et al. Exp Mol Med. 2004，36(6):576-81. [2] Dedeoglu A，et al. J Neurosci. 2002，22(20):8942-50. |
| Unit | Bottle |
| Specification | 50mg 100mg |
Remark：These protocols are for reference only. Solarbio does not independently validate these methods.
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1. The products are all for scientific research use only. Do not use it for medical, clinical diagnosis or treatment, food and cosmetics, etc. Do not store them in ordinary residential areas.
2. For your safety and health, please wear laboratory clothes, disposable gloves and masks.
3. The experimental results may be affected by many factors, after-sale service is limited to the product itself and does not involve other compensation.
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